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C5-benzyl SAHA
CAS No. 2115700-64-4
C5-benzyl SAHA ( —— )
产品货号. M13367 CAS No. 2115700-64-4
C5-benzyl SAHA is a C5-modified SAHA analog that displays dual selectivity to HDAC.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 100MG | 获取报价 | 有现货 |
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| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称C5-benzyl SAHA
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述C5-benzyl SAHA is a C5-modified SAHA analog that displays dual selectivity to HDAC.
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产品描述C5-benzyl SAHA is a C5-modified SAHA analog that displays dual selectivity to HDAC6 (IC50=0.27 uM) and HDAC8 (IC50=0.38 uM) over HDAC 1, 2, and 3 (IC50=2.9-5.8 uM); dose dependently and selectively increases in levels of acetyl-α-tubulin in U937 leukemia cells.
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同义词——
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通路Cell Cycle/DNA Damage
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靶点HDAC
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受体HDAC
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研究领域——
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适应症——
化学信息
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CAS Number2115700-64-4
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分子量354.45
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分子式C21H26N2O3
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纯度>98% (HPLC)
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溶解度——
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SMILES——
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化学全称4-benzyl-N8-hydroxy-N1-phenyloctanediamide
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Negmeldin AT, et al. Bioorg Med Chem Lett. 2017 Aug 1;27(15):3254-3258.
产品手册
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